The synthesis and receptor binding affinities of DDD-016, a novel, potential, atypical antipsychotic

Achintya K. Bandyopadhyaya, Desikan R Rajagopalan, Nigam Rath, Amy Herrold, Raghavan Rajagopalan, T. Celesete Napier, Clark E. Tedford, Parthasarathi Rajagopalan

Research output: Contribution to journalArticlepeer-review

Abstract

A new pentacyclic compound, DDD-016 (10d) was designed and synthesized as a potential antipsychotic and screened for binding affinity in a broad panel of over 80 CNS and other receptors, monoamine transporters, and ion channels. The resulting receptor binding profile of DDD-016 is consistent with that of an improved atypical antipsychotic candidate.
Original languageAmerican English
JournalMedChemComm
Volume3
DOIs
StatePublished - May 7 2012

Disciplines

  • Life Sciences
  • Biochemistry, Biophysics, and Structural Biology
  • Biochemistry

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